SCHEMBL8769869

SCHEMBL8769869

NC(F)(F)C(F)(F)C(F)(F)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.56
PTPN5 P54829 1/20 0.46
CYP2C9 P11712 1/20 0.39
TAAR1 Q96RJ0 2/20 0.39
CYP3A4 P08684 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
BACE1 P56817 1/20 0.39
ALDH1A1 P00352 3/20 0.38
AKT1 P31749 1/20 0.37
AKT2 P31751 1/20 0.37
PTPN1 P18031 1/20 0.36
KCNN4 O15554 1/20 0.36
TSHR P16473 1/20 0.36
KDM1A O60341 2/20 0.35
MAOB P27338 1/20 0.35
GLO1 Q04760 1/20 0.35
DGAT1 O75907 1/20 0.35
KCNH2 Q12809 1/20 0.35
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669394 0.83 KIF11 (0.60) KIF11PTPN5CYP2C9TAAR1CYP3A4
SCHEMBL1421311 0.79 KIF11 (0.56) KIF11PTPN5CYP2C9TAAR1CYP3A4
SCHEMBL16439869 0.78 KIF11 (0.65) KIF11PTPN5CYP2C9TAAR1CYP3A4
SCHEMBL25808753 0.78 KIF11 (0.65) KIF11PTPN5CYP2C9TAAR1CYP3A4
Biphenyl SCHEMBL28313556 0.74 ALDH1A1 (0.60) KIF11PTPN5TAAR1CYP3A4HSD17B10
Hydrazine SCHEMBL27541145 0.73 KIF11 (0.90) KIF11PTPN5BACE1ALDH1A1TSHR
SCHEMBL28070215 0.72 KIF11 (0.56) KIF11PTPN5CYP2C9TAAR1CYP3A4
SCHEMBL9579980 0.72 KCNN4 (0.52) KIF11TAAR1ALDH1A1PTPN1KCNN4
SCHEMBL163728 0.72 KIF11 (1.00) KIF11PTPN5BACE1ALDH1A1TSHR
SCHEMBL25013355 0.72 KIF11 (0.47) KIF11PTPN5CYP2C9TDP1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793671-A1 PHENYLSUBSTITUTED 4-AZASTEROID FLUORODERIVATIVES PHARMACIA & UPJOHN S.p.A. (IT) 1997-09-10 EP disclosed
WO-1997010257-A1 PHENYLSUBSTITUTED 4-AZASTEROID FLUORODERIVATIVES PHARMACIA & UPJOHN S.P.A. (IT) 1997-03-20 WO disclosed