SCHEMBL669394

SCHEMBL669394

FC(F)(F)C(F)(F)C(F)(F)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.60
PTPN5 P54829 3/20 0.48
CYP2C9 P11712 1/20 0.42
BACE1 P56817 1/20 0.41
ALDH1A1 P00352 3/20 0.41
TSHR P16473 1/20 0.39
PTPN1 P18031 2/20 0.38
MAPK1 P28482 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MMP3 P08254 1/20 0.37
BCL2L1 Q07817 1/20 0.37
GLO1 Q04760 1/20 0.37
DGAT1 O75907 1/20 0.37
KCNH2 Q12809 1/20 0.37
SCN2A Q99250 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1421311 0.91 KIF11 (0.56) KIF11PTPN5CYP2C9BACE1ALDH1A1
SCHEMBL25808753 0.86 KIF11 (0.65) KIF11PTPN5CYP2C9BACE1ALDH1A1
SCHEMBL16439869 0.86 KIF11 (0.65) KIF11PTPN5CYP2C9BACE1ALDH1A1
SCHEMBL11696796 0.85 TSHR (0.52) KIF11PTPN5ALDH1A1TSHRPTPN1
SCHEMBL8769869 0.83 KIF11 (0.56) KIF11PTPN5CYP2C9BACE1ALDH1A1
Biphenyl SCHEMBL6131233 0.81 ALDH1A1 (0.48) KIF11PTPN5CYP2C9BACE1ALDH1A1
SCHEMBL3390346 0.78 TSHR (0.50) KIF11PTPN5ALDH1A1TSHRPTPN1
SCHEMBL10453463 0.76 TSHR (0.48) KIF11PTPN5ALDH1A1TSHRPTPN1
SCHEMBL9800786 0.76 TSHR (0.48) KIF11PTPN5ALDH1A1TSHRPTPN1
SCHEMBL15320774 0.76 TSHR (0.48) KIF11PTPN5ALDH1A1TSHRPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9758453-B2 One-component reagent for the fluoroalkylation reaction THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2017-09-12 US disclosed
US-9758453-B2 One-component reagent for the fluoroalkylation reaction THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2017-09-12 US disclosed
US-20160185691-A1 One-Component Reagent for the Fluoroalkylation Reaction THE BOARD OF TRUSTEES OF THE UNIVERSITY OF LLLINOIS (US) 2016-06-30 US disclosed
US-20160185691-A1 One-Component Reagent for the Fluoroalkylation Reaction THE BOARD OF TRUSTEES OF THE UNIVERSITY OF LLLINOIS (US) 2016-06-30 US disclosed
US-9193648-B2 Fluoroalkylation methods and reagents BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2015-11-24 US disclosed
US-9193648-B2 Fluoroalkylation methods and reagents BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2015-11-24 US disclosed
US-20130225815-A1 Fluoroalkylation Methods And Reagents THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2013-08-29 US disclosed
US-20130225815-A1 Fluoroalkylation Methods And Reagents THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2013-08-29 US disclosed
EP-2606048-A1 FLUOROALKYLATION METHODS AND REAGENTS The Board of Trustees of the University of Illinois (US) 2013-06-26 EP disclosed
WO-2012024564-A1 FLUOROALKYLATION METHODS AND REAGENTS THE BOARD OF TRUSTESS OF THE UNIVERSITY OF ILLINOIS (US) 2012-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130225815-A1 Fluoroalkylation Methods And Reagents ALK, AFF4, AFF2 KIF11 2064/4885PTPN5 934/4885CYP2C9 772/4885
US-20160185691-A1 One-Component Reagent for the Fluoroalkylation Reaction AOC1, AOC3, AOC2 KIF11 1521/4885PTPN5 2214/4885CYP2C9 930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.