SCHEMBL8770103

SCHEMBL8770103

CS(=O)(=O)c1cccc(-c2ccc(Br)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.49
NR1H2 P55055 8/20 0.48
NR1H3 Q13133 3/20 0.47
CA12 O43570 2/20 0.46
CA2 P00918 2/20 0.46
CA9 Q16790 2/20 0.46
ALDH1A1 P00352 1/20 0.45
MAPK1 P28482 1/20 0.45
PTGS2 P35354 3/20 0.43
GRIA2 P42262 1/20 0.43
KIF11 P52732 1/20 0.42
RXRA P19793 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6243674 0.86 KCNH2 (0.50) KCNH2NR1H2NR1H3PTGS2LOXL2
SCHEMBL29321413 0.85 ALDH1A1 (0.48) KCNH2NR1H2NR1H3CA12CA2
SCHEMBL2140712 0.84 PTGS2 (0.53) KCNH2NR1H2NR1H3ALDH1A1PTGS2
SCHEMBL15758712 0.82 CYP19A1 (0.60) CA12CA2CA9ALDH1A1
SCHEMBL14320650 0.81 CA12 (0.51) KCNH2NR1H2NR1H3CA12CA2
SCHEMBL5831675 0.81 PTGS2 (0.56) NR1H2NR1H3PTGS2
SCHEMBL17153735 0.81 PTGS2 (0.50) KCNH2NR1H2NR1H3CA12CA2
SCHEMBL5893176 0.81 NR1H2 (0.51) KCNH2NR1H2NR1H3LOXL2
SCHEMBL5908704 0.80 CA2 (0.61) CA12CA2CA9PTGS2KIF11
SCHEMBL21770154 0.79 CA12 (0.53) KCNH2NR1H2NR1H3CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0794942-A1 SUBSTITUTED BIPHENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-09-17 EP disclosed
WO-1996016934-A1 SUBSTITUTED BIPHENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-06-06 WO disclosed