SCHEMBL8771387

SCHEMBL8771387

Nc1ccc(Cl)cc1C(=O)NCCN1CCCC1

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.61
HTR4 Q13639 2/20 0.58
EPHX2 P34913 1/20 0.57
CYP2C19 P33261 1/20 0.54
CNR1 P21554 1/20 0.53
GAA P10253 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
CACNA1G O43497 2/20 0.51
CCR2 P41597 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8771374 0.89 CYP2C19 (0.69) ALDH1A1EPHX2CYP2C19SMN1; SMN2
SCHEMBL9410255 0.82 ALDH1A1 (0.59) ALDH1A1HTR4EPHX2CYP2C19CNR1
SCHEMBL26758003 0.81 LMNA (0.60) ALDH1A1HTR4CYP2C19SMN1; SMN2
SCHEMBL27985765 0.81 ALDH1A1 (0.62) ALDH1A1HTR4
SCHEMBL11554175 0.80 CYP2C19 (0.81) ALDH1A1EPHX2CYP2C19SMN1; SMN2
SCHEMBL11277010 0.80 KDM4E (0.61) ALDH1A1HTR4
SCHEMBL3543948 0.79 ALDH1A1 (0.65) ALDH1A1HTR4SMN1; SMN2CACNA1G
SCHEMBL10705234 0.79 CDK1 (0.57) ALDH1A1
SCHEMBL7813262 0.77 RECQL (0.68) ALDH1A1CNR1
SCHEMBL19359526 0.77 TNKS (0.50) ALDH1A1CYP2C19CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620218-B1 2, 3-Dihydro-4(1H)-quinazolinones active in gastro-intestinal pathologies ALFA WASSERMANN SPA (IT) 1997-10-01 EP disclosed
US-5446152-A Antiemetic agent ALFA WASSERMANN S.P.A. (IT) 1995-08-29 US disclosed
EP-0620218-A1 Heterocyclic compounds active in gastro-intestinal pathologies ALFA WASSERMANN S.p.A. (IT) 1994-10-19 EP disclosed