SCHEMBL8771705

SCHEMBL8771705

COC(=O)c1ccc(C(=O)Nc2ccc3c(c2)C(c2ccccc2)=CC3(C)C)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.55
KMT2A Q03164 3/20 0.53
CTDSP1 Q9GZU7 1/20 0.53
RAB9A P51151 4/20 0.50
RARB P10826 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
KDM4E B2RXH2 3/20 0.50
RARA P10276 2/20 0.50
RARG P13631 2/20 0.50
MEN1 O00255 2/20 0.50
LMNA P02545 2/20 0.50
MAPT P10636 2/20 0.50
PKM P14618 2/20 0.47
TRPV1 Q8NER1 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
NPC1 O15118 3/20 0.45
ATM Q13315 1/20 0.45
ALDH1A1 P00352 2/20 0.44
TP53 P04637 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8771636 0.93 RARA (0.58) PTPN1KMT2ACTDSP1RAB9ARARB
SCHEMBL8771889 0.90 RARA (0.61) KMT2ARAB9ARARBRARARARG
SCHEMBL8771689 0.86 PDK2 (0.49) PTPN1KMT2ARAB9ARARBRARA
SCHEMBL27462421 0.84 RARA (0.72) PTPN1KMT2ACTDSP1RAB9ARARB
SCHEMBL4653413 0.83 RARA (0.71) KMT2ARARBKDM4ERARARARG
SCHEMBL8771880 0.82 RARA (0.55) PTPN1KMT2ARAB9ARARBRARA
SCHEMBL8771890 0.82 RARA (0.55) PTPN1KMT2ARAB9ARARBRARA
SCHEMBL8771810 0.78 KMT2A (0.48) KMT2ARAB9ASMN1; SMN2KDM4EMEN1
SCHEMBL17275573 0.75 RARB (0.50) KMT2ARARBRARARARGALDH1A1
SCHEMBL22223650 0.75 PTPN1 (0.94) PTPN1KMT2ARAB9ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661259-B1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL MYERS SQUIBB CO (US) 1997-10-08 EP disclosed
US-5648385-A TREATING RHEUMATOID ARTHRITIS BRISTOL-MYERS SQUIBB CO. (US) 1997-07-15 US disclosed
US-5618839-A Retinoid-like compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1997-04-08 US disclosed
CN-1144217-A Retinoid-like compounds BRISTOL MYERS SQUIBB CO (US) 1997-03-05 CN disclosed
EP-0661259-A1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL-MYERS SQUIBB COMPANY (US) 1995-07-05 EP disclosed