SCHEMBL877180

SCHEMBL877180

CC(C)n1nc(-c2ccc(NC(=O)c3cc4cccnc4s3)cc2)cc1C(=O)NCCN1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.43
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
JAK2 O60674 5/20 0.42
ATR Q13535 4/20 0.42
FLT3 P36888 2/20 0.41
SYK P43405 2/20 0.41
CHRNA7 P36544 2/20 0.41
HDAC6 Q9UBN7 1/20 0.41
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
KCNH2 Q12809 1/20 0.39
JAK3 P52333 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
IKBKG Q9Y6K9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL876612 0.84 CHRNA7 (0.46) NAMPTCHRNA7HDAC6
SCHEMBL877181 0.83 NAMPT (0.40) NAMPTDRD2DRD3JAK2CHRNA7
SCHEMBL874515 0.83 ATR (0.43) NAMPTDRD2DRD3JAK2ATR
SCHEMBL874686 0.80 CYP3A4 (0.42) NAMPTDRD2DRD3JAK2ATR
SCHEMBL873657 0.79 CYP3A4 (0.41) NAMPTDRD2DRD3JAK2ATR
SCHEMBL874535 0.79 NAMPT (0.48) NAMPTDRD2DRD3JAK2ATR
SCHEMBL873820 0.79 ATR (0.46) NAMPTDRD2DRD3JAK2ATR
SCHEMBL874058 0.78 NAMPT (0.42) NAMPTDRD2DRD3JAK2ATR
SCHEMBL875500 0.78 ATR (0.41) NAMPTDRD2DRD3JAK2ATR
SCHEMBL873629 0.78 NAMPT (0.42) NAMPTDRD2DRD3JAK2ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed