SCHEMBL874535

SCHEMBL874535

O=C(NCCN1CCCCC1)c1ccc(-c2ccc(NC(=O)c3cc4cccnc4s3)cc2)o1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.48
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
ATR Q13535 3/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
KCNH2 Q12809 1/20 0.40
CHRNA7 P36544 1/20 0.40
IKBKB O14920 1/20 0.40
CHUK O15111 1/20 0.40
IKBKG Q9Y6K9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873905 0.94 DRD2 (0.48) NAMPTDRD2DRD3ALDH1A1KCNH2
SCHEMBL874022 0.91 CHRNA7 (0.41) NAMPTDRD2DRD3ALDH1A1KDM4E
SCHEMBL874135 0.90 NAMPT (0.41) NAMPTDRD2DRD3ALDH1A1KDM4E
SCHEMBL873709 0.89 CHRNA7 (0.41) NAMPTDRD2DRD3ALDH1A1KDM4E
SCHEMBL873865 0.85 NAMPT (0.42) NAMPTALDH1A1KDM4ENPC1GAA
SCHEMBL873871 0.83 NPC1 (0.42) NAMPTALDH1A1KDM4ENPC1GAA
SCHEMBL874184 0.81 NPC1 (0.41) NAMPTALDH1A1KDM4ENPC1GAA
SCHEMBL874187 0.81 NPC1 (0.46) ALDH1A1KDM4ENPC1GAAHPGD
SCHEMBL874536 0.81 NAMPT (0.45) NAMPTALDH1A1KDM4ENPC1GAA
SCHEMBL874617 0.81 DRD2 (0.44) NAMPTDRD2DRD3ATRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed