SCHEMBL874058

SCHEMBL874058

CCNc1cc(-c2ccc(NC(=O)c3cc4cccnc4s3)cc2)ccc1C(=O)NCCN1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.42
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
JAK2 O60674 3/20 0.39
ATR Q13535 3/20 0.39
CHRNA7 P36544 3/20 0.39
WNT1 P04628 1/20 0.39
DYRK1A Q13627 1/20 0.39
BRAF P15056 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
KCNH2 Q12809 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874686 0.88 CYP3A4 (0.42) NAMPTDRD2DRD3JAK2ATR
SCHEMBL873657 0.84 CYP3A4 (0.41) NAMPTDRD2DRD3JAK2ATR
SCHEMBL874059 0.84 NAMPT (0.41) NAMPTDRD2DRD3CHRNA7MKNK2
SCHEMBL874339 0.83 MKNK1 (0.39) NAMPTCHRNA7DYRK1ACYP3A4NPSR1
SCHEMBL874515 0.82 ATR (0.43) NAMPTDRD2DRD3JAK2ATR
SCHEMBL874015 0.81 DRD2 (0.41) NAMPTDRD2DRD3CHRNA7KCNH2
SCHEMBL873820 0.81 ATR (0.46) NAMPTDRD2DRD3JAK2ATR
SCHEMBL875500 0.80 ATR (0.41) NAMPTDRD2DRD3JAK2ATR
SCHEMBL874151 0.80 CYP3A4 (0.40) NAMPTDRD2DRD3ATRCHRNA7
SCHEMBL874535 0.80 NAMPT (0.48) NAMPTDRD2DRD3JAK2ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed