SCHEMBL8771832

SCHEMBL8771832

CC1(C)CCC(=O)c2cc(S)ccc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.33
ALDH1A1 P00352 3/20 0.33
HIF1A Q16665 2/20 0.33
EPAS1 Q99814 2/20 0.33
KDM4E B2RXH2 2/20 0.33
LMNA P02545 2/20 0.33
POLB P06746 2/20 0.33
RECQL P46063 2/20 0.33
HSD17B10 Q99714 2/20 0.33
MEN1 O00255 1/20 0.33
CES2 O00748 1/20 0.33
APAF1 O14727 1/20 0.33
TERT O14746 1/20 0.33
EED O75530 1/20 0.33
MAPT P10636 1/20 0.33
AKR1B1 P15121 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
CES1 P23141 1/20 0.33
APEX1 P27695 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6992256 0.81 ALDH1A1 (0.42) TP53ALDH1A1HIF1AEPAS1KDM4E
SCHEMBL31650524 0.79 PBRM1 (0.53) ALDH1A1KDM4ELMNAMAPTESR1
SCHEMBL6240700 0.79 HSD17B10 (0.44) TP53ALDH1A1HIF1AEPAS1KDM4E
SCHEMBL8662092 0.79 PBRM1 (0.53) ALDH1A1KDM4ELMNAMAPTESR1
SCHEMBL8662369 0.79 TDP2 (0.40) TP53ALDH1A1HIF1AEPAS1KDM4E
SCHEMBL15716876 0.79 MALT1 (0.41) ALDH1A1POLBMAPTCES1RXRA
SCHEMBL30279114 0.79 MALT1 (0.41) MEN1CES1KMT2ATDP1L3MBTL1
SCHEMBL445935 0.79 MALT1 (0.41) MEN1CES1KMT2ATDP1L3MBTL1
SCHEMBL18856493 0.78 ALDH1A1 (0.34) TP53ALDH1A1HIF1AEPAS1KDM4E
SCHEMBL2061344 0.77 KDM4E (0.45) ALDH1A1KDM4EMAPK1CYP3A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661259-B1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL MYERS SQUIBB CO (US) 1997-10-08 EP disclosed
US-5648385-A TREATING RHEUMATOID ARTHRITIS BRISTOL-MYERS SQUIBB CO. (US) 1997-07-15 US disclosed
US-5618839-A Retinoid-like compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1997-04-08 US disclosed
EP-0661259-A1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL-MYERS SQUIBB COMPANY (US) 1995-07-05 EP disclosed