SCHEMBL8771897

SCHEMBL8771897

CC1(C)CCC(=O)c2cc(O[Si](C)(C)C(C)(C)C)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.43
CA1 P00915 4/20 0.43
CA9 Q16790 4/20 0.43
PREP P48147 3/20 0.39
GRM2 Q14416 1/20 0.32
RXRA P19793 3/20 0.32
RXRB P28702 2/20 0.32
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32
RXRG P48443 1/20 0.32
MALT1 Q9UDY8 2/20 0.31
PPARG P37231 2/20 0.30
PRNP P04156 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
CES2 O00748 1/20 0.30
APAF1 O14727 1/20 0.30
TERT O14746 1/20 0.30
EED O75530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4786577 0.79 CA12 (0.48) CA12CA1CA9PREP
SCHEMBL31650634 0.79 KDM4E (0.45) CA1CA9MALT1PRNPKDM4E
SCHEMBL2061344 0.79 KDM4E (0.45) CA1CA9MALT1PRNPKDM4E
SCHEMBL4517231 0.78 RXRA (0.32) PREPRXRAPPARGKDM4EMEN1
SCHEMBL7566980 0.77 MAOA (0.50) CA12CA1CA9PREPMEN1
SCHEMBL6280495 0.76 RXRA (0.36) RXRARXRBRARARARBRARG
SCHEMBL6280497 0.75 PPARG (0.41) PPARGMAPTKMT2A
SCHEMBL31650617 0.74 RXRA (0.37) RXRARXRBRARARARBRARG
SCHEMBL24529065 0.73 MAOB (0.48) CA12CA1CA9PREPHSD17B10
SCHEMBL445935 0.72 MALT1 (0.41) CA1CA9MALT1MEN1CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661259-B1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL MYERS SQUIBB CO (US) 1997-10-08 EP disclosed
US-5648385-A TREATING RHEUMATOID ARTHRITIS BRISTOL-MYERS SQUIBB CO. (US) 1997-07-15 US disclosed
US-5618839-A Retinoid-like compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1997-04-08 US disclosed
EP-0661259-A1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL-MYERS SQUIBB COMPANY (US) 1995-07-05 EP disclosed