SCHEMBL8772633

SCHEMBL8772633

C#Cc1c(C(=O)O)cccc1-c1ccc2c(c1)C(C)(C)CC=C2c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RARB P10826 18/20 0.47
RARG P13631 18/20 0.47
RARA P10276 17/20 0.47
RXRA P19793 2/20 0.45
NR2E1 Q9Y466 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8772796 0.94 RARB (0.48) RARBRARGRARARXRANR2E1
SCHEMBL8772837 0.84 RARA (0.35) RARBRARGRARA
SCHEMBL8772745 0.84 RARA (0.50) RARBRARGRARARXRA
SCHEMBL8772773 0.84 RARA (0.39) RARBRARGRARARXRA
SCHEMBL8772664 0.81 RARB (0.40) RARBRARGRARARXRANR2E1
SCHEMBL8772662 0.80 RARB (0.42) RARBRARGRARARXRANR2E1
SCHEMBL8772764 0.80 RARB (0.33) RARBRARGRARARXRA
SCHEMBL8562392 0.79 RARB (0.42) RARBRARGRARARXRA
SCHEMBL8772736 0.78 RARB (0.38) RARBRARGRARARXRANR2E1
SCHEMBL8772826 0.77 RARB (0.39) RARBRARGRARARXRANR2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800517-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1997-10-15 EP disclosed