SCHEMBL8772745

SCHEMBL8772745

C#Cc1c(C(=O)O)cccc1-c1ccc2c(c1)C(C)(C)CC=C2C#Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RARA P10276 17/20 0.50
RARB P10826 17/20 0.42
RARG P13631 17/20 0.42
RXRA P19793 1/20 0.36
HNF4A P41235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8772773 0.90 RARA (0.39) RARARARBRARGRXRA
SCHEMBL8772633 0.84 RARB (0.47) RARARARBRARGRXRA
SCHEMBL8772662 0.81 RARB (0.42) RARARARBRARGRXRA
SCHEMBL8772796 0.80 RARB (0.48) RARARARBRARGRXRA
SCHEMBL8772664 0.78 RARB (0.40) RARARARBRARGRXRA
SCHEMBL8772741 0.78 RARA (0.53) RARARARBRARGHNF4A
SCHEMBL8772736 0.77 RARB (0.38) RARARARBRARGRXRA
SCHEMBL8772764 0.77 RARB (0.33) RARARARBRARGRXRA
SCHEMBL8562392 0.76 RARB (0.42) RARARARBRARGRXRA
SCHEMBL8772837 0.75 RARA (0.35) RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800517-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1997-10-15 EP disclosed