SCHEMBL8772649

SCHEMBL8772649

CC1(C)CC=Cc2ccc(Br)cc21

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.31
HTR2C P28335 1/20 0.30
BACE1 P56817 2/20 0.30
HIF1A Q16665 1/20 0.30
EPAS1 Q99814 1/20 0.30
CMA1 P23946 1/20 0.30
AHR P35869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026331 0.87 HIF1A (0.33) HTR2CBACE1HIF1AEPAS1CMA1
SCHEMBL9485242 0.84 KDM1A (0.30) KDM1A
SCHEMBL30659806 0.78 AKR1B1 (0.33) KDM1AHTR2CHIF1AEPAS1
SCHEMBL8031290 0.77 TDP2 (0.36) HIF1AEPAS1
SCHEMBL7604066 0.75 SIGMAR1 (0.40) HTR2C
SCHEMBL8170079 0.73 HIF1A (0.33) HIF1AEPAS1
SCHEMBL30320303 0.72 HIF1A (0.33) HIF1AEPAS1
SCHEMBL4369386 0.72 HIF1A (0.33) HIF1AEPAS1
SCHEMBL869051 0.72 IDO1 (0.34)
SCHEMBL26105726 0.72 NQO1 (0.31) HIF1AEPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997048672-A2 SUBSTITUTED TETRAHYDRONAPHTHALENE AND DIHYDRONAPHTHALENE DERIVATIVES HAVING RETINOID AND/OR RETINOID ANTAGONIST-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 1997-12-24 WO disclosed
EP-0800517-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1997-10-15 EP disclosed