SCHEMBL8772741

SCHEMBL8772741

CC1(C)CC=C(C#Cc2ccccc2)c2ccc(C#Cc3ccccc3C(=O)O)cc21

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RARA P10276 17/20 0.53
RARB P10826 16/20 0.48
RARG P13631 16/20 0.48
HNF4A P41235 1/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
CYP26A1 O43174 1/20 0.41
CYP3A4 P08684 1/20 0.41
CRABP2 P29373 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8772769 0.93 RARA (0.45) RARARARBRARGCYP26A1CYP3A4
SCHEMBL7637516 0.86 RARA (0.68) RARARARBRARGCYP26A1CYP3A4
SCHEMBL8772626 0.85 RARA (0.62) RARARARBRARG
SCHEMBL8772660 0.82 RARA (0.53) RARARARBRARGCYP26A1CYP3A4
SCHEMBL8772792 0.81 RARB (0.61) RARARARBRARG
SCHEMBL8772762 0.79 RARA (0.41) RARARARBRARGHNF4ACYP26A1
SCHEMBL7637426 0.78 RARA (0.52) RARARARBRARGCYP26A1CYP3A4
SCHEMBL8772745 0.78 RARA (0.50) RARARARBRARGHNF4A
SCHEMBL7640578 0.77 RARA (0.58) RARARARBRARGCYP26A1CYP3A4
SCHEMBL7806999 0.77 RARA (0.78) RARARARBRARGCYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800517-A1 ACETYLENES DISUBSTITUTED WITH A 5 OR 8 SUBSTITUTED TETRAHYDRONAPHTHYL OR DIHYDRONAPHTHYL GROUP AND WITH AN ARYL OR HETEROARYL GROUPS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1997-10-15 EP disclosed