SCHEMBL8773594

SCHEMBL8773594

CCN(CC)CCCP(c1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.50
KCNH2 Q12809 5/20 0.48
SLC6A4 P31645 4/20 0.48
SLC6A2 P23975 3/20 0.48
CHRM1 P11229 2/20 0.48
ADRA1A P35348 2/20 0.48
OPRM1 P35372 2/20 0.48
DRD3 P35462 2/20 0.48
SLC6A3 Q01959 2/20 0.48
CHRM2 P08172 1/20 0.48
HTR1A P08908 1/20 0.48
ADRA2A P08913 1/20 0.48
DRD1 P21728 1/20 0.48
HRH1 P35367 2/20 0.41
DRD2 P14416 1/20 0.41
ADRA2C P18825 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
OPRK1 P41145 1/20 0.41
MTOR P42345 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9619532 0.88 SIGMAR1 (0.44) SIGMAR1KCNH2SLC6A4SLC6A2CHRM1
SCHEMBL10733880 0.86 SIGMAR1 (0.43) SIGMAR1KCNH2SLC6A4SLC6A2CHRM1
SCHEMBL8723759 0.85 SIGMAR1 (0.42) SIGMAR1KCNH2SLC6A4SLC6A2CHRM1
SCHEMBL2879292 0.84 KCNH2 (0.47) SIGMAR1KCNH2SLC6A4SLC6A2CHRM1
SCHEMBL4659134 0.80 HTR2A (0.47) SIGMAR1KCNH2SLC6A4SLC6A2CHRM1
SCHEMBL30626104 0.80 TDP1 (0.33) KCNH2SLC6A4SLC6A2CHRM1ADRA1A
SCHEMBL5033519 0.79 MEN1 (0.45) KCNH2SLC6A4SLC6A2CHRM1ADRA1A
Propane SCHEMBL17007613 0.79 TDP1 (0.39) KCNH2SLC6A4SLC6A2CHRM1ADRA1A
SCHEMBL19753210 0.79 KDM4E (0.40) SIGMAR1KCNH2SLC6A4SLC6A2CHRM1
Hydrochloric Acid SCHEMBL10947305 0.79 KCNH2 (0.49) SIGMAR1KCNH2OPRM1DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696304-A REACTING CONJUGATED ALKADIENOL WITH WATER USING PALLADIUM CATALYST IN LOW BOILING REACTION SOLVENT, THEN DISTILLATION MITSUBISHI CHEMICAL CORPORATION (JP) 1997-12-09 US disclosed
EP-0605735-B1 PROCESS FOR PRODUCING ALKADIENOL MITSUBISHI CHEM CORP (JP) 1997-11-05 EP disclosed
US-5557016-A HYDROXYLATION OF CONJUGATED ALKADIENES IN THE PRESENCE OF PALLADIUM CATALYSIS MITSUBISHI KASEI CORPORATION (JP) 1996-09-17 US disclosed
EP-0361304-B1 Method for producing alkadienols MITSUBISHI CHEM CORP (JP) 1996-02-21 EP disclosed
EP-0605735-A1 PROCESS FOR PRODUCING ALKADIENOL Mitsubishi Chemical Corporation (JP) 1994-07-13 EP disclosed
US-4990698-A Method for producing alkadienols MITSUBISHI KASEI CORPORATION (JP) 1991-02-05 US disclosed
EP-0361304-A2 Method for producing alkadienols Mitsubishi Chemical Corporation (JP) 1990-04-04 EP disclosed
US-4687874-A Selective hydroformylation process using alkyl diaryl phosphine rhodium carbonyl hydride catalysts EXXON RESEARCH AND ENGINEERING COMPANY (US) 1987-08-18 US disclosed
US-4687866-A Ligand exchange process for producing alkyl diaryl phosphine rhodium carbonyl hydrides EXXON RESEARCH AND ENGINEERING COMPANY (US) 1987-08-18 US disclosed
US-4668809-A ALKYL DIARYLPHOSPHINE RHODIUM CARBONYL HYDRIDES, HYDROFORMYLATION, OLEFINS EXXON RESEARCH AND ENGINEERING (US) 1987-05-26 US disclosed
US-4595753-A Nitrogen heterocycle substituted EXXON RESEARCH AND ENGINEERING CO. (US) 1986-06-17 US disclosed
EP-0024091-B1 HYDROFORMYLATION PROCESS AND NOVEL TRANSITION METAL CATALYSTS EXXON RESEARCH AND ENGINEERING COMPANY (US) 1985-04-03 EP disclosed
EP-0024091-A4 HYDROFORMYLATION PROCESS AND NOVEL TRANSITION METAL CATALYSTS. EXXON RESEARCH ENGINEERING CO (US) 1981-07-16 EP disclosed
EP-0024091-A1 HYDROFORMYLATION PROCESS AND NOVEL TRANSITION METAL CATALYSTS. EXXON RESEARCH ENGINEERING CO (US) 1981-02-25 EP disclosed
WO-1980001690-A1 CARBONYLATION PROCESS AND NOVEL TRANSITION METAL CATALYSTS EXXON RESEARCH ENGINEERING CO (US) 1980-08-21 WO disclosed