SCHEMBL877377

SCHEMBL877377

COC(=O)c1cc(-c2ccc(C)cc2)n(-c2ccc(S)cc2)n1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 2/20 0.58
SMN1; SMN2 Q16637 3/20 0.57
PTGS2 P35354 2/20 0.57
PPP1CA P62136 1/20 0.57
CA9 Q16790 1/20 0.56
RPA1 P27694 3/20 0.52
MALT1 Q9UDY8 2/20 0.49
NFKB1 P19838 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
MAPK9 P45984 1/20 0.48
CHRNA7 P36544 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14728116 0.94 SMPD1 (0.64) SMPD1SMN1; SMN2PTGS2PPP1CACA9
SCHEMBL878349 0.86 SMN1; SMN2 (0.76) SMPD1SMN1; SMN2PPP1CARPA1
SCHEMBL3866686 0.85 SMPD1 (0.56) SMPD1SMN1; SMN2PTGS2PPP1CACA9
SCHEMBL16797379 0.84 KDM1A (0.60) SMPD1SMN1; SMN2PTGS2PPP1CACA9
SCHEMBL861458 0.84 SMPD1 (0.55) SMPD1SMN1; SMN2PTGS2PPP1CACA9
SCHEMBL13290381 0.84 PTGS2 (0.66) SMPD1SMN1; SMN2PTGS2PPP1CACA9
SCHEMBL3863977 0.84 PTGS2 (0.66) SMPD1SMN1; SMN2PTGS2PPP1CACA9
SCHEMBL14728144 0.83 SMPD1 (0.54) SMPD1SMN1; SMN2PTGS2PPP1CACA9
SCHEMBL3874092 0.83 PTGS2 (0.82) SMN1; SMN2PTGS2CA9MAPK9CHRNA7
SCHEMBL8369157 0.83 RPA1 (0.65) SMPD1SMN1; SMN2PTGS2PPP1CACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143302-B2 Methods and compositions for diagnostic and therapeutic targeting of COX-2 VANDERBILT UNIVERSITY (US) 2012-03-27 US disclosed
US-20100254910-A1 METHODS AND COMPOSITIONS FOR DIAGNOSTIC AND THERAPEUTIC TARGETING OF COX-2 VANDERBILT UNIVERSITY (US) 2010-10-07 US disclosed
US-7736624-B2 derivatives of non-steroidal anti-inflammatory drugs that exhibit selective binding to cyclooxygenase-2 (COX-2) and that comprise functional groups allowing them to be used for medical diagnosis and/or as therapeutic agents; tissue-targeted therapy UNIV VANDERBILT (US) 2010-06-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100254910-A1 METHODS AND COMPOSITIONS FOR DIAGNOSTIC AND THERAPEUTIC TARGETING OF COX-2 PTGS2, PTGES2, PTGER2 SMPD1 677/4885SMN1; SMN2 1445/4885PTGS2 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.