SCHEMBL8774349

SCHEMBL8774349

NC(=O)Nc1ccc2cn[nH]c2c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.67
CYP1A2 P05177 2/20 0.67
CYP3A4 P08684 2/20 0.67
CYP2D6 P10635 2/20 0.67
CYP2C9 P11712 2/20 0.67
HIF1A Q16665 2/20 0.67
HSD17B10 Q99714 2/20 0.67
CYP2C19 P33261 1/20 0.67
PHLPP2 Q6ZVD8 1/20 0.67
CLK2 P49760 2/20 0.62
CLK4 Q9HAZ1 2/20 0.62
MAP4K4 O95819 1/20 0.62
DYRK1A Q13627 1/20 0.62
SRPK1 Q96SB4 1/20 0.62
HPGD P15428 3/20 0.60
MAPT P10636 9/20 0.59
KDM4E B2RXH2 8/20 0.59
RAB9A P51151 3/20 0.59
NPC1 O15118 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30026503 1.00 ALDH1A1 (0.67) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL30933139 0.87 ROCK2 (0.72) ALDH1A1CLK2CLK4MAP4K4DYRK1A
SCHEMBL5225654 0.87 ROCK2 (0.72) ALDH1A1CLK2CLK4MAP4K4DYRK1A
SCHEMBL1548213 0.85 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL30725947 0.85 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL14045319 0.84 ROCK2 (0.77) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5823003 0.84 ALDH1A1 (0.77) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL23084047 0.80 HPGD (0.63) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL21688513 0.80 ROCK1 (0.79) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL22590423 0.80 ALDH1A1 (0.61) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0804425-A2 BENZODIAZEPINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-05 EP disclosed