SCHEMBL8774747

SCHEMBL8774747

CCc1ccc(-c2cnc(F)c(F)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.42
METAP2 P50579 1/20 0.39
CYP17A1 P05093 3/20 0.38
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
TP53 P04637 3/20 0.37
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
GRM5 P41594 2/20 0.36
GPR55 Q9Y2T6 1/20 0.36
CYP3A4 P08684 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35
GRIN2B Q13224 3/20 0.35
GRIN1 Q05586 1/20 0.35
LMNA P02545 1/20 0.35
CHRNA7 P36544 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8775015 1.00 EGLN1 (0.42) EGLN1METAP2CYP17A1CYP11B1CYP11B2
SCHEMBL8774798 0.88 FEN1 (0.40) EGLN1
SCHEMBL8775052 0.86 RAB9A (0.48) CYP17A1CYP11B1CYP11B2TP53NPC1
SCHEMBL8774871 0.86 RAB9A (0.48) CYP17A1CYP11B1CYP11B2TP53NPC1
SCHEMBL8774132 0.85 NPC1 (0.40) EGLN1METAP2CYP17A1CYP11B1TP53
SCHEMBL8774800 0.83 RARB (0.49) TP53NPC1PKMRAB9ASMN1; SMN2
SCHEMBL8774086 0.83 RARB (0.49) TP53NPC1PKMRAB9ASMN1; SMN2
SCHEMBL8774269 0.82 RARB (0.55) NPC1RAB9ASMN1; SMN2HSD17B10
SCHEMBL8774355 0.82 RARB (0.55) NPC1RAB9ASMN1; SMN2HSD17B10
SCHEMBL8774259 0.81 FEN1 (0.40) NPC1RAB9ASMN1; SMN2GRIN2BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed