SCHEMBL8774768

SCHEMBL8774768

CCCCCOc1ccc(-c2cnc(Cl)c(Cl)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HSD17B10 Q99714 1/20 0.54
CYP2D6 P10635 9/20 0.51
CYP3A4 P08684 6/20 0.51
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 2/20 0.49
HTT P42858 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CYP2C9 P11712 6/20 0.49
CYP2C19 P33261 6/20 0.49
CYP19A1 P11511 5/20 0.49
RARB P10826 3/20 0.48
CYP1A2 P05177 3/20 0.47
NR5A1 Q13285 1/20 0.45
LTA4H P09960 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774531 0.99 NPC1 (0.52) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6
SCHEMBL8774496 0.91 RAB9A (0.49) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6
SCHEMBL8876334 0.86 NPC1 (0.51) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6
SCHEMBL8877313 0.86 NPC1 (0.51) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6
SCHEMBL8875742 0.86 NPC1 (0.51) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6
SCHEMBL8774722 0.84 ALDH1A1 (0.53) NPC1RAB9AKDM4EALDH1A1L3MBTL1
SCHEMBL6499085 0.81 THRB (0.43) NPC1RAB9ASMN1; SMN2HSD17B10KDM4E
SCHEMBL7185520 0.81 NPC1 (0.62) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6
SCHEMBL8774115 0.81 RAB9A (0.49) NPC1RAB9ASMN1; SMN2HSD17B10KDM4E
SCHEMBL9160256 0.80 NPC1 (0.58) NPC1RAB9ASMN1; SMN2HSD17B10CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed