SCHEMBL8774912

SCHEMBL8774912

CCCCc1ccc(-c2ccc(C#Cc3cc(F)c(F)nc3F)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.43
HSD17B10 Q99714 1/20 0.43
FFAR1 O14842 3/20 0.40
RARB P10826 4/20 0.40
RARA P10276 1/20 0.40
RARG P13631 1/20 0.40
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
PTPN11 Q06124 1/20 0.35
PTPRO Q16827 1/20 0.35
HSD11B1 P28845 1/20 0.35
GPR84 Q9NQS5 1/20 0.35
CTRC Q99895 1/20 0.35
EIF4A1 P60842 2/20 0.35
NISCH Q9Y2I1 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
NFKB1 P19838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774909 0.96 HSD17B10 (0.48) TSHRHSD17B10FFAR1RARBRARA
SCHEMBL8774821 0.96 FFAR1 (0.43) TSHRHSD17B10FFAR1RARBRARA
SCHEMBL8774374 0.92 FFAR1 (0.42) TSHRHSD17B10FFAR1RARBRARA
SCHEMBL8774994 0.92 FFAR1 (0.42) TSHRHSD17B10FFAR1RARBRARA
SCHEMBL8774302 0.91 HSD17B10 (0.43) TSHRHSD17B10FFAR1RARBRARA
SCHEMBL8774295 0.88 FFAR1 (0.44) FFAR1S1PR1
SCHEMBL8774750 0.87 FFAR1 (0.38) FFAR1RARBRARARARGNPC1
SCHEMBL8775170 0.85 CYP2D6 (0.46) HSD17B10RARBRARANPC1RAB9A
SCHEMBL8774468 0.85 FFAR1 (0.40) TSHRHSD17B10FFAR1PTPN11PTPRO
SCHEMBL31633923 0.84 TSHR (0.47) TSHRHSD17B10FFAR1RARBRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed