SCHEMBL8774750

SCHEMBL8774750

CCc1ccc(-c2ccc(C#Cc3cc(F)c(F)nc3F)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 6/20 0.38
CYP2A6 P11509 1/20 0.35
ACACB O00763 3/20 0.33
EGLN1 Q9GZT9 1/20 0.33
FFAR4 Q5NUL3 1/20 0.32
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32
GRM5 P41594 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
FAAH O00519 1/20 0.30
GCGR P47871 1/20 0.30
MAPK14 Q16539 1/20 0.30
NPC1 O15118 1/20 0.30
POLB P06746 1/20 0.30
GAA P10253 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774297 0.96 FFAR1 (0.40) FFAR1CYP2A6ACACBEGLN1FFAR4
SCHEMBL8774994 0.89 FFAR1 (0.42) FFAR1ACACBFFAR4RARARARB
SCHEMBL8774912 0.87 TSHR (0.43) FFAR1RARARARBRARGSMN1; SMN2
SCHEMBL8774909 0.85 HSD17B10 (0.48) FFAR1RARARARBRARGSMN1; SMN2
SCHEMBL8774295 0.84 FFAR1 (0.44) FFAR1ACACBFFAR4
SCHEMBL8775031 0.83 CYP11B1 (0.39) FFAR1ACACBFFAR4SMN1; SMN2NPC1
SCHEMBL8774403 0.83 FFAR1 (0.38) FFAR1CYP2A6ACACBEGLN1FFAR4
SCHEMBL8774821 0.82 FFAR1 (0.43) FFAR1FFAR4RARARARBRARG
SCHEMBL8774463 0.81 MCHR1 (0.41) ACACBSMN1; SMN2NPC1GAARAB9A
SCHEMBL8775170 0.81 CYP2D6 (0.46) RARARARBSMN1; SMN2NPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed