SCHEMBL8775100

SCHEMBL8775100

CCCCC1CCC(C(C)c2ccc(-c3cnc(F)c(F)c3)cc2)CC1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.33
GRIN2B Q13224 6/20 0.32
GRIN1 Q05586 2/20 0.32
PTGS2 P35354 4/20 0.32
PDE5A O76074 1/20 0.32
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
MAPK1 P28482 1/20 0.31
KMT2A Q03164 1/20 0.31
GPR55 Q9Y2T6 1/20 0.31
TP53 P04637 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30
CDK7 P50613 1/20 0.30
CDK13 Q14004 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774704 0.97 PDE5A (0.33) ESR2GRIN2BGRIN1PTGS2PDE5A
SCHEMBL8774698 0.96 GAA (0.33) ESR2GRIN2BGRIN1PTGS2PDE5A
SCHEMBL8774654 0.96 GAA (0.33) ESR2GRIN2BGRIN1PTGS2PDE5A
SCHEMBL8774394 0.93 GRIN2B (0.33) GRIN2BGRIN1PTGS2GPR55CDK7
SCHEMBL8774169 0.88 GRIN2B (0.36) GRIN2BGRIN1PTGS2GPR55CDK7
SCHEMBL9155759 0.85 PTGS2 (0.35) PTGS2MEN1GAAMAPK1KMT2A
SCHEMBL8774317 0.83 SLC6A2 (0.35) PTGS2MEN1GAAMAPK1KMT2A
SCHEMBL8774509 0.82 CYP2C9 (0.38) ESR2GRIN2BGRIN1PDE5AMEN1
SCHEMBL8775102 0.82 RARB (0.38) ESR2GRIN2BGRIN1PDE5AMEN1
SCHEMBL8775108 0.82 RARB (0.38) ESR2GRIN2BGRIN1PDE5AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed