SCHEMBL8774169

SCHEMBL8774169

CCC1CCC(C(C)c2ccc(-c3cnc(F)c(F)c3)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 7/20 0.36
GRIN1 Q05586 4/20 0.36
ALOX5AP P20292 2/20 0.35
FEN1 P39748 2/20 0.35
PTGS2 P35354 4/20 0.34
GPR55 Q9Y2T6 2/20 0.33
CDK7 P50613 1/20 0.32
CDK13 Q14004 1/20 0.32
CYP17A1 P05093 1/20 0.32
ACACB O00763 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TRPV3 Q8NET8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774394 0.90 GRIN2B (0.33) GRIN2BGRIN1PTGS2GPR55CDK7
SCHEMBL8775100 0.88 ESR2 (0.33) GRIN2BGRIN1PTGS2GPR55CDK7
SCHEMBL8774704 0.87 PDE5A (0.33) GRIN2BGRIN1PTGS2GPR55
SCHEMBL8774654 0.86 GAA (0.33) GRIN2BGRIN1PTGS2GPR55
SCHEMBL8774698 0.86 GAA (0.33) GRIN2BGRIN1PTGS2GPR55
SCHEMBL9158975 0.83 PTGS2 (0.37) PTGS2
SCHEMBL8775244 0.81 SLC6A2 (0.38) GRIN2BGRIN1PTGS2ACACB
SCHEMBL8774117 0.81 DGAT1 (0.39) GRIN2BGRIN1ALOX5APFEN1GPR55
SCHEMBL8774122 0.81 DGAT1 (0.39) GRIN2BGRIN1ALOX5APFEN1GPR55
SCHEMBL8774613 0.80 TRPV3 (0.37) TRPV3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed