SCHEMBL8776264

SCHEMBL8776264

O=C(CCC1CC[CH]CC1)N1CCN(c2ccnnc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 2/20 0.46
HIF1A Q16665 1/20 0.46
ADAMTS5 Q9UNA0 2/20 0.43
TP53 P04637 1/20 0.42
POLB P06746 2/20 0.41
LMNA P02545 3/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MMP2 P08253 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KMT2A Q03164 1/20 0.39
MAPK1 P28482 1/20 0.38
ADAMTS4 O75173 1/20 0.38
HTR1A P08908 1/20 0.38
HTR7 P34969 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7790314 0.86 ALDH1A1 (0.47) ALDH1A1KDM4EMAPTHIF1AADAMTS5
SCHEMBL7790836 0.79 ITGB3 (0.46) ALDH1A1KDM4EMAPTHIF1ALMNA
SCHEMBL7790329 0.77 MAPT (0.50) ALDH1A1KDM4EMAPTHIF1ALMNA
SCHEMBL7787452 0.76 KDM4E (0.46) ALDH1A1KDM4EMAPTLMNANPSR1
SCHEMBL7790323 0.72 MAPT (0.52) ALDH1A1KDM4EMAPTHIF1ALMNA
SCHEMBL7790305 0.71 ITGB3 (0.47) ALDH1A1KDM4E
SCHEMBL7790309 0.71 ITGB3 (0.57) ALDH1A1KDM4EMAPTHIF1ALMNA
SCHEMBL8355447 0.70 POLB (0.38) ALDH1A1KDM4EMAPTHIF1AADAMTS5
SCHEMBL7787422 0.70 TDP1 (0.49) ALDH1A1MAPTKMT2A
SCHEMBL7791932 0.68 ITGB3 (0.52) ALDH1A1KDM4EMAPTHIF1AMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808311-A2 NEW DERIVATIVES OF PYRIDIL PIPERAZINE OR PYRIDAZINYL PIPERAZYL, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1997-11-26 EP disclosed
WO-1996024581-A2 DERIVATIVES OF PYRIDIL PIPERAZINE OR PYRIDAZINYL PIPERAZYL, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1996-08-15 WO disclosed