SCHEMBL8776633

SCHEMBL8776633

COC(=O)CN(C(C)=O)C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.58
CHRM2 P08172 5/20 0.56
CHRM3 P20309 5/20 0.56
ACHE P22303 3/20 0.52
SIGMAR1 Q99720 2/20 0.52
DRD2 P14416 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
HTR2B P41595 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9057752 0.99 OPRM1 (0.57) OPRM1CHRM2CHRM3ACHESIGMAR1
Hydrochloric Acid SCHEMBL9024089 0.87 OPRM1 (0.56) OPRM1CHRM2CHRM3ACHESIGMAR1
Hydrochloric Acid SCHEMBL8480640 0.84 OPRM1 (0.52) OPRM1CHRM2CHRM3SIGMAR1DRD2
Hydrochloric Acid SCHEMBL8486085 0.84 LTA4H (0.58) OPRM1CHRM2CHRM3ACHESIGMAR1
SCHEMBL9653759 0.81 OPRM1 (0.65) OPRM1CHRM2CHRM3ACHESIGMAR1
SCHEMBL14839622 0.79 OPRM1 (0.55) OPRM1CHRM2CHRM3ACHESIGMAR1
SCHEMBL9030647 0.78 SIGMAR1 (0.67) OPRM1CHRM2CHRM3ACHESIGMAR1
SCHEMBL9653783 0.77 OPRM1 (0.57) OPRM1CHRM2CHRM3ACHESIGMAR1
Hydrochloric Acid SCHEMBL8480247 0.77 SIGMAR1 (0.53) OPRM1CHRM2CHRM3ACHESIGMAR1
SCHEMBL9471497 0.77 SIGMAR1 (0.62) OPRM1CHRM2CHRM3ACHESIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799202-A1 PIPERAZINE DERIVATIVES, MEDICAMENTS CONTAINING THE SAME, THEIR USE AND PROCESS FOR PREPARING THE SAME Dr. Karl Thomae GmbH (DE) 1997-10-08 EP disclosed