SCHEMBL8776765

SCHEMBL8776765

CCS(=O)(=O)c1ccc(-c2cc(C#N)c(OCc3ccc(OC)cc3)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 15/20 0.60
CNR2 P34972 4/20 0.45
PTGS2 P35354 2/20 0.44
PTGS1 P23219 1/20 0.44
SQOR Q9Y6N5 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
ABHD6 Q9BV23 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101056 0.92 CNR1 (0.61) CNR1CNR2PTGS2PTGS1SQOR
SCHEMBL8093740 0.91 CNR1 (0.60) CNR1CNR2PTGS2PTGS1SQOR
SCHEMBL8776720 0.87 PTGS2 (0.47) CNR1CNR2PTGS2PTGS1SQOR
SCHEMBL8095103 0.86 CNR1 (0.61) CNR1CNR2PTGS2PTGS1
SCHEMBL8086461 0.84 CNR1 (0.61) CNR1CNR2PTGS2PTGS1
SCHEMBL8086096 0.82 CNR1 (0.69) CNR1CNR2PTGS2PTGS1
SCHEMBL8776822 0.81 PTGS2 (0.56) CNR1CNR2PTGS2PTGS1SQOR
SCHEMBL8086786 0.81 CNR1 (0.64) CNR1PTGS2PTGS1
SCHEMBL8101395 0.81 CNR1 (0.55) CNR1CNR2PTGS2PTGS1
SCHEMBL8095797 0.80 CNR1 (0.69) CNR1CNR2PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed