SCHEMBL8776720

SCHEMBL8776720

CCS(=O)(=O)c1ccc(-c2cc(C#N)c(OC)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.47
PTGS1 P23219 1/20 0.47
SQOR Q9Y6N5 7/20 0.46
CNR1 P21554 7/20 0.45
CNR2 P34972 1/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SCN9A Q15858 1/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8776770 0.90 SCN9A (0.45) SQORCNR1CNR2SCN9AKDM4E
SCHEMBL215205 0.89 PTGS2 (0.53) PTGS2PTGS1SQORCNR1CNR2
SCHEMBL8776778 0.89 CNR1 (0.41) PTGS2PTGS1SQORCNR1CNR2
SCHEMBL8093195 0.88 PTGS2 (0.47) PTGS2PTGS1SQORCNR1CNR2
SCHEMBL7055227 0.87 SQOR (0.46) PTGS2PTGS1SQORCNR1CNR2
SCHEMBL8776765 0.87 CNR1 (0.60) PTGS2PTGS1SQORCNR1CNR2
SCHEMBL8776866 0.86 KDM4E (0.43) PTGS2CNR1CNR2MEN1KMT2A
SCHEMBL8776822 0.86 PTGS2 (0.56) PTGS2PTGS1SQORCNR1CNR2
SCHEMBL8776749 0.84 PTGS2 (0.47) PTGS2PTGS1CNR1CNR2NPSR1
SCHEMBL8776752 0.83 CNR1 (0.48) SQORCNR1CNR2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed