SCHEMBL8776835

SCHEMBL8776835

CS(=O)(=O)c1[c]c(-c2ccc(F)cc2)ccc1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 0.45
PTGS1 P23219 6/20 0.41
NR3C1 P04150 1/20 0.37
PGR P06401 1/20 0.37
NR3C2 P08235 1/20 0.37
AR P10275 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6930665 0.85 PTGS2 (0.36) PTGS2PTGS1
SCHEMBL9119298 0.84 PTGS2 (0.38) PTGS2PTGS1
SCHEMBL5030910 0.84 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL9118988 0.83 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL9117197 0.83 PLCG1 (0.37) PTGS2
SCHEMBL7505306 0.83 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL9119397 0.80 EGFR (0.38) PTGS2PTGS1NR3C1
SCHEMBL9118873 0.80 PTGS2 (0.42) PTGS2PTGS1
SCHEMBL9116829 0.79 PTGS2 (0.43) PTGS2
SCHEMBL3822120 0.77 NPC1 (0.36) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO claimed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed
WO-1995030652-A1 SUBSTITUTED SPIRODIENES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed