SCHEMBL877703

SCHEMBL877703

CC(C)Nc1nc(Cl)ccc1C(=O)NCCN1CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
NPSR1 Q6W5P4 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
HTR4 Q13639 1/20 0.47
HSD17B10 Q99714 1/20 0.47
POLB P06746 1/20 0.46
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
HPGD P15428 1/20 0.45
KMT2A Q03164 1/20 0.45
HRH3 Q9Y5N1 1/20 0.44
GLA P06280 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL485925 0.86 ALDH1A1 (0.48) ALDH1A1NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL11977016 0.75 LMNA (0.73) ALDH1A1NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL12015824 0.74 LMNA (0.75) ALDH1A1NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL1758196 0.73 ALDH1A1 (0.65) ALDH1A1NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL21883951 0.73 MEN1 (0.52) ALDH1A1NPSR1CYP1A2CYP2D6CYP2C9
SCHEMBL2740260 0.73 MEN1 (0.53) ALDH1A1NPSR1POLBMEN1KMT2A
SCHEMBL21883952 0.72 NPSR1 (0.52) ALDH1A1NPSR1POLBMEN1KMT2A
SCHEMBL15636352 0.72 MAPT (0.45) ALDH1A1KDM4EMEN1KMT2AL3MBTL1
SCHEMBL15296616 0.71 NPSR1 (0.61) ALDH1A1NPSR1HTR4HSD17B10MEN1
SCHEMBL15495475 0.71 ALDH1A1 (0.54) ALDH1A1NPSR1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed