SCHEMBL8777069

SCHEMBL8777069

NCCc1ccccc1Oc1ccccc1CO

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.65
TAAR1 Q96RJ0 8/20 0.58
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
HTR2A P28223 3/20 0.41
CXCL8 P10145 2/20 0.41
MPO P05164 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2A6 P11509 1/20 0.38
NFKB1 P19838 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR2C P28335 1/20 0.38
HTR7 P34969 1/20 0.38
CTSK P43235 1/20 0.38
HTR6 P50406 1/20 0.38
CYP2A13 Q16696 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6311971 0.90 HRH1 (0.77) HRH1TAAR1HTR2ACXCL8CYP2A6
SCHEMBL5950358 0.85 SLC6A2 (0.50) HRH1SLC6A2SLC6A4CXCL8
SCHEMBL8777062 0.84 HRH1 (0.44) HRH1TAAR1SLC6A2SLC6A4CXCL8
SCHEMBL11100370 0.84 HRH1 (0.44) HRH1TAAR1SLC6A2SLC6A4CXCL8
SCHEMBL10862161 0.79 TAAR1 (0.67) HRH1TAAR1HTR2AMPOCYP1A2
SCHEMBL2356168 0.78 CXCL8 (0.64) SLC6A2SLC6A4CXCL8
SCHEMBL1569927 0.78 HRH1 (1.00) HRH1TAAR1SLC6A2SLC6A4HTR2A
Hydrochloric Acid SCHEMBL10862159 0.77 TAAR1 (0.64) HRH1TAAR1HTR2AMPOCYP1A2
SCHEMBL6236000 0.77 HRH1 (0.48) HRH1TAAR1SLC6A2SLC6A4CXCL8
SCHEMBL8777076 0.77 HRH1 (0.50) HRH1TAAR1SLC6A2SLC6A4CXCL8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800513-A1 OPIATE RECEPTOR LIGANDS CHIRON CORPORATION (US) 1997-10-15 EP disclosed
US-5605932-A Opiate receptor ligands CHIRON CORPORATION (US) 1997-02-25 US disclosed
US-5536868-A Opiate receptor ligands CHIRON CORPORATION (US) 1996-07-16 US disclosed
WO-1996020921-A1 OPIATE RECEPTOR LIGANDS CHIRON CORPORATION (US) 1996-07-11 WO disclosed
US-5481020-A Opiate receptor ligands CHIRON CORPORATION (US) 1996-01-02 US disclosed