SCHEMBL8777076

SCHEMBL8777076

NCc1ccccc1Oc1ccccc1CCO

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.50
TAAR1 Q96RJ0 2/20 0.44
DPP4 P27487 1/20 0.39
CXCL8 P10145 2/20 0.38
PNMT P11086 1/20 0.38
AOC3 Q16853 1/20 0.36
SLC6A4 P31645 4/20 0.36
SLC6A2 P23975 3/20 0.36
TDP1 Q9NUW8 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
BRD4 O60885 1/20 0.34
RIPK1 Q13546 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6236000 0.90 HRH1 (0.48) HRH1TAAR1CXCL8AOC3SLC6A4
SCHEMBL6319190 0.85 HRH1 (0.52) HRH1TAAR1DPP4CXCL8PNMT
SCHEMBL8777062 0.84 HRH1 (0.44) HRH1TAAR1DPP4CXCL8PNMT
SCHEMBL11100370 0.84 HRH1 (0.44) HRH1TAAR1CXCL8SLC6A4SLC6A2
SCHEMBL28327254 0.79 TAAR1 (0.52) TAAR1AOC3SLC6A4SLC6A2SLC6A3
SCHEMBL632593 0.79 DPP4 (0.48) TAAR1DPP4PNMTTDP1
SCHEMBL1067253 0.78 HRH1 (0.67) HRH1SLC6A4SLC6A2TDP1SLC6A3
SCHEMBL17024100 0.78 HRH1 (0.46) HRH1TAAR1CXCL8SLC6A4SLC6A2
SCHEMBL5694864 0.78 TAAR1 (0.44) HRH1TAAR1AOC3TDP1HTR1A
SCHEMBL6311971 0.77 HRH1 (0.77) HRH1TAAR1CXCL8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800513-A1 OPIATE RECEPTOR LIGANDS CHIRON CORPORATION (US) 1997-10-15 EP disclosed
US-5605932-A Opiate receptor ligands CHIRON CORPORATION (US) 1997-02-25 US disclosed
US-5536868-A Opiate receptor ligands CHIRON CORPORATION (US) 1996-07-16 US disclosed
WO-1996020921-A1 OPIATE RECEPTOR LIGANDS CHIRON CORPORATION (US) 1996-07-11 WO disclosed
US-5481020-A Opiate receptor ligands CHIRON CORPORATION (US) 1996-01-02 US disclosed