SCHEMBL8777097

SCHEMBL8777097

CC(NC(=O)[C@H]1CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C)C(O)C(F)(F)F

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.64
CYP3A4 P08684 6/20 0.64
ALDH1A1 P00352 6/20 0.64
MAPT P10636 6/20 0.64
LMNA P02545 6/20 0.64
MAPK1 P28482 4/20 0.64
TSHR P16473 3/20 0.64
SHBG P04278 3/20 0.64
SERPINA6 P08185 3/20 0.64
CYP2C9 P11712 2/20 0.64
HIF1A Q16665 2/20 0.64
ABCB11 O95342 2/20 0.64
KDM4E B2RXH2 2/20 0.64
NR3C2 P08235 2/20 0.64
MEN1 O00255 2/20 0.64
NR3C1 P04150 2/20 0.64
PGR P06401 2/20 0.64
AR P10275 2/20 0.64
KMT2A Q03164 2/20 0.64
GPBAR1 Q8TDU6 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9110297 1.00 SMN1; SMN2 (0.64) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA
SCHEMBL8994150 0.84 SRD5A2 (0.62) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA
SCHEMBL8994147 0.84 SRD5A2 (0.62) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA
SCHEMBL9402957 0.84 CYP3A4 (0.68) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA
SCHEMBL9402948 0.84 CYP3A4 (0.68) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA
SCHEMBL9109527 0.83 ALDH1A1 (0.53) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA
SCHEMBL9109519 0.83 ALDH1A1 (0.53) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA
SCHEMBL8634489 0.83 SRD5A2 (0.75) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA
SCHEMBL4986169 0.82 CYP3A4 (0.78) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA
SCHEMBL8994121 0.82 LMNA (0.68) SMN1; SMN2CYP3A4ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0611374-B1 17-BETA-SUBSTITUTED 4-AZA-5-ALPHA-ANDROSTAN-3-ONE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 1997-10-22 EP disclosed
EP-0681587-A1 SIDE CHAIN FLUORO SUBSTITUTED 3-CARBOXYSTEROIDS PHARMACIA & UPJOHN S.p.A. (IT) 1995-11-15 EP disclosed
WO-1995014709-A1 SIDE CHAIN FLUORO SUBSTITUTED 3-CARBOXYSTEROIDS PHARMACIA S.P.A. (IT) 1995-06-01 WO disclosed
US-5418238-A 17β-substituted 4-aza-5α-androstan-3-one derivatives FARMITALIA CARLO ERBA S.R.L. (IT) 1995-05-23 US disclosed