SCHEMBL8779017

SCHEMBL8779017

O=C1c2ccc(OCc3ccccc3)cc2CCC12CCCC2

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 18/20 0.63
MAOA P21397 17/20 0.63
KDM1A O60341 1/20 0.49
TOP1 P11387 1/20 0.49
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
NFKB1 P19838 1/20 0.48
GRM5 P41594 1/20 0.48
RAB9A P51151 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30769168 0.99 MAOB (0.65) MAOBMAOAKDM1ANPC1ALDH1A1
SCHEMBL8778993 0.90 MAOB (0.63) MAOBMAOAKDM1ATOP1NPC1
SCHEMBL8778979 0.85 MAOA (0.56) MAOBMAOAKDM1A
SCHEMBL1359950 0.85 MAOB (0.62) MAOBMAOAKDM1ATOP1NPC1
SCHEMBL30769243 0.81 MAOB (0.60) MAOBMAOAKDM1ATOP1NPC1
SCHEMBL30769325 0.81 MAOB (0.57) MAOBMAOAKDM1ATOP1NPC1
SCHEMBL30768524 0.79 MAOA (0.59) MAOBMAOAKDM1A
SCHEMBL226640 0.78 MAOB (1.00) MAOBMAOANPC1ALDH1A1HPGD
SCHEMBL3451690 0.78 MAOB (0.94) MAOBMAOANPC1ALDH1A1HPGD
SCHEMBL8778973 0.78 MAOA (0.56) MAOBMAOAKDM1ATOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0606661-B1 Octahydrophenanthrene derivatives and their use as NMDA-Antagonists HOFFMANN LA ROCHE (CH) 1997-03-12 EP disclosed
US-5385947-A For prevention of nerve damage due to reduction of blood or oxygen supplies HOFFMANN-LA ROCHE INC. (US) 1995-01-31 US disclosed
EP-0606661-A1 Octahydrophenanthrene derivatives and their use as NMDA-Antagonists F. HOFFMANN-LA ROCHE AG (CH) 1994-07-20 EP disclosed