SCHEMBL8778979

SCHEMBL8778979

C=C1c2ccc(OCc3ccccc3)cc2CCC12CCCC2

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOA P21397 11/20 0.56
MAOB P27338 11/20 0.56
KDM1A O60341 2/20 0.49
HRH3 Q9Y5N1 4/20 0.46
CYP2D6 P10635 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8778973 0.90 MAOA (0.56) MAOAMAOBKDM1AHRH3CYP2D6
SCHEMBL8779017 0.85 MAOB (0.63) MAOAMAOBKDM1A
SCHEMBL30769168 0.84 MAOB (0.65) MAOAMAOBKDM1A
SCHEMBL8778993 0.78 MAOB (0.63) MAOAMAOBKDM1AHRH3
SCHEMBL17355183 0.75 MAOB (0.53) MAOAMAOBKDM1AHRH3
SCHEMBL1359950 0.74 MAOB (0.62) MAOAMAOBKDM1AHRH3
SCHEMBL8779163 0.73 HTT (0.46) MAOAMAOB
SCHEMBL8778939 0.73 MAPT (0.41) KDM1A
SCHEMBL226640 0.72 MAOB (1.00) MAOAMAOB
SCHEMBL3451690 0.72 MAOB (0.94) MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0606661-B1 Octahydrophenanthrene derivatives and their use as NMDA-Antagonists HOFFMANN LA ROCHE (CH) 1997-03-12 EP disclosed
US-5385947-A For prevention of nerve damage due to reduction of blood or oxygen supplies HOFFMANN-LA ROCHE INC. (US) 1995-01-31 US disclosed
EP-0606661-A1 Octahydrophenanthrene derivatives and their use as NMDA-Antagonists F. HOFFMANN-LA ROCHE AG (CH) 1994-07-20 EP disclosed