SCHEMBL8779030

SCHEMBL8779030

O=C1c2cc(Cl)c(Cl)cc2CCC12CCCC2

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 13/20 0.39
HTR2A P28223 11/20 0.39
HTR2C P28335 11/20 0.39
HTR2B P41595 11/20 0.39
DRD2 P14416 11/20 0.39
KDM1A O60341 1/20 0.34
TYMS P04818 1/20 0.34
PDE7A Q13946 1/20 0.32
CES1 P23141 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779094 0.79 SIGMAR1 (0.57) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL8779128 0.79 F7 (0.46) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL8778969 0.79 KDM1A (0.34) KDM1A
SCHEMBL9588126 0.76 KDM1A (0.35) KDM1ATYMSCES1
SCHEMBL8779154 0.72 PARP1 (0.46) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL8779110 0.72 SIGMAR1 (0.43) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL8779101 0.72 TDP1 (0.50) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL8778995 0.72 SIGMAR1 (0.43) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL22892512 0.72 SIGMAR1 (0.46) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL8778968 0.72 MEN1 (0.36) SIGMAR1HTR2AHTR2CHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0606661-B1 Octahydrophenanthrene derivatives and their use as NMDA-Antagonists HOFFMANN LA ROCHE (CH) 1997-03-12 EP disclosed
US-5385947-A For prevention of nerve damage due to reduction of blood or oxygen supplies HOFFMANN-LA ROCHE INC. (US) 1995-01-31 US disclosed
EP-0606661-A1 Octahydrophenanthrene derivatives and their use as NMDA-Antagonists F. HOFFMANN-LA ROCHE AG (CH) 1994-07-20 EP disclosed