SCHEMBL8778968

SCHEMBL8778968

O=C1c2cc(Cl)cc(Cl)c2CCC12CCCC2

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NOTUM Q6P988 1/20 0.35
ADRA2A P08913 1/20 0.35
CES1 P23141 2/20 0.35
DNMT1 P26358 1/20 0.35
PDE7A Q13946 1/20 0.35
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
SIGMAR1 Q99720 2/20 0.32
DRD2 P14416 1/20 0.32
SPR P35270 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779032 0.84 AR (0.33) MEN1KMT2AL3MBTL1CES1DNMT1
SCHEMBL8779104 0.80 ADRA2A (0.35) NOTUMADRA2A
SCHEMBL8779031 0.77 SIGMAR1 (0.40) L3MBTL1NOTUMCES1PDE7AHTR2A
SCHEMBL8779128 0.73 F7 (0.46) PDE7AHTR2AHTR2CHTR2BSIGMAR1
SCHEMBL8779030 0.72 SIGMAR1 (0.39) CES1PDE7AHTR2AHTR2CHTR2B
SCHEMBL8779094 0.70 SIGMAR1 (0.57) HTR2AHTR2CHTR2BSIGMAR1DRD2
SCHEMBL7815325 0.69 MEN1 (0.49) MEN1KMT2AL3MBTL1NOTUMCES1
SCHEMBL29844266 0.69 MEN1 (0.52) MEN1KMT2AL3MBTL1NOTUMCES1
SCHEMBL2256507 0.69 MEN1 (0.52) MEN1KMT2AL3MBTL1NOTUMCES1
SCHEMBL28000654 0.66 MEN1 (0.49) MEN1KMT2AL3MBTL1NOTUMCES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0606661-B1 Octahydrophenanthrene derivatives and their use as NMDA-Antagonists HOFFMANN LA ROCHE (CH) 1997-03-12 EP disclosed
US-5385947-A For prevention of nerve damage due to reduction of blood or oxygen supplies HOFFMANN-LA ROCHE INC. (US) 1995-01-31 US disclosed
EP-0606661-A1 Octahydrophenanthrene derivatives and their use as NMDA-Antagonists F. HOFFMANN-LA ROCHE AG (CH) 1994-07-20 EP disclosed