SCHEMBL8779208

SCHEMBL8779208

CC(C)CCOc1ccnc(OC(=O)NC(=O)[C@@H](N)C(C)C)c1O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.38
GALR3 O60755 1/20 0.33
HSP90AA1 P07900 1/20 0.33
EPHX2 P34913 1/20 0.33
CYP19A1 P11511 1/20 0.33
XDH P47989 1/20 0.32
MAPK1 P28482 1/20 0.32
KDM4E B2RXH2 1/20 0.31
PPIA P62937 1/20 0.31
TLR8 Q9NR97 1/20 0.31
MCHR1 Q99705 1/20 0.31
CARM1 Q86X55 1/20 0.31
PRMT6 Q96LA8 1/20 0.31
GRM2 Q14416 1/20 0.31
CIT O14578 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779278 0.91 HTT (0.39) HTTGALR3HSP90AA1EPHX2CYP19A1
SCHEMBL8779223 0.88 AAK1 (0.39) HTTCIT
SCHEMBL8779253 0.84 HTT (0.39) HTTGALR3HSP90AA1EPHX2CYP19A1
SCHEMBL8779210 0.84 CIT (0.30) CIT
SCHEMBL8779418 0.83 PPARG (0.36) MCHR1
SCHEMBL8883147 0.82 HTT (0.39) HTTGALR3HSP90AA1EPHX2CYP19A1
SCHEMBL8779325 0.81 IKBKB (0.37) MAPK1KDM4ECARM1PRMT6
SCHEMBL8779136 0.81 IKBKB (0.37) MAPK1KDM4ECARM1PRMT6
SCHEMBL8779135 0.80 XIAP (0.40) CARM1PRMT6
SCHEMBL8779157 0.80 XIAP (0.40) CARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed