SCHEMBL8779136

SCHEMBL8779136

CCCOc1ccnc(OC(=O)NC(=O)[C@H](C)N)c1O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.37
XIAP P98170 1/20 0.36
CARM1 Q86X55 2/20 0.36
PRMT6 Q96LA8 2/20 0.36
HSD17B10 Q99714 2/20 0.34
MAPT P10636 2/20 0.34
SLC15A1 P46059 1/20 0.33
ACACB O00763 6/20 0.32
MAPK1 P28482 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779325 1.00 IKBKB (0.37) IKBKBXIAPCARM1PRMT6HSD17B10
SCHEMBL8779135 0.94 XIAP (0.40) XIAPCARM1PRMT6SLC15A1ACACB
SCHEMBL8779157 0.94 XIAP (0.40) XIAPCARM1PRMT6SLC15A1ACACB
SCHEMBL8779165 0.93 XIAP (0.38) XIAPCARM1PRMT6MAPTSLC15A1
SCHEMBL8779212 0.91 HPGD (0.38) IKBKBCARM1PRMT6KDM4EALDH1A1
SCHEMBL8779176 0.91 HPGD (0.38) IKBKBCARM1PRMT6KDM4EALDH1A1
SCHEMBL8779278 0.90 HTT (0.39) CARM1PRMT6ACACBMAPK1KDM4E
SCHEMBL8779183 0.89 REN (0.35) IKBKBCARM1PRMT6ACACB
SCHEMBL8779140 0.89 REN (0.35) IKBKBCARM1PRMT6ACACB
SCHEMBL8779292 0.87 CARM1 (0.35) CARM1PRMT6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed