SCHEMBL8779157

SCHEMBL8779157

CCCCOc1ccnc(OC(=O)NC(=O)[C@H](C)N)c1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.40
SLC15A1 P46059 1/20 0.37
CARM1 Q86X55 2/20 0.36
PRMT6 Q96LA8 2/20 0.36
LMNA P02545 4/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
FAAH O00519 5/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
STAT3 P40763 1/20 0.34
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
ACACB O00763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779135 1.00 XIAP (0.40) XIAPSLC15A1CARM1PRMT6LMNA
SCHEMBL8779165 0.97 XIAP (0.38) XIAPSLC15A1CARM1PRMT6LMNA
SCHEMBL8779136 0.94 IKBKB (0.37) XIAPSLC15A1CARM1PRMT6LMNA
SCHEMBL8779325 0.94 IKBKB (0.37) XIAPSLC15A1CARM1PRMT6LMNA
SCHEMBL8779183 0.90 REN (0.35) CARM1PRMT6ACACB
SCHEMBL8779140 0.90 REN (0.35) CARM1PRMT6ACACB
SCHEMBL8779212 0.90 HPGD (0.38) CARM1PRMT6LMNASMN1; SMN2
SCHEMBL8779176 0.90 HPGD (0.38) CARM1PRMT6LMNASMN1; SMN2
SCHEMBL8779278 0.89 HTT (0.39) CARM1PRMT6ACACB
SCHEMBL8779292 0.86 CARM1 (0.35) CARM1PRMT6SMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed