SCHEMBL8779657

SCHEMBL8779657

Cc1cc(C=C2CCN(C(N)=O)C2=O)cc(C)c1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.55
EEF2K O00418 1/20 0.42
SRC P12931 1/20 0.42
AKR1B1 P15121 1/20 0.40
MEN1 O00255 2/20 0.38
LMNA P02545 2/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
CYP1A2 P05177 4/20 0.37
CYP3A4 P08684 4/20 0.37
CYP2B6 P20813 3/20 0.37
CYP2D6 P10635 1/20 0.37
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
XBP1 P17861 1/20 0.35
MPI P34949 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779651 1.00 CYP2C9 (0.55) CYP2C9EEF2KSRCAKR1B1MEN1
SCHEMBL8779655 0.83 CYP1A2 (0.58) CYP2C9EEF2KSRCMEN1KMT2A
SCHEMBL8779659 0.83 CYP1A2 (0.58) CYP2C9EEF2KSRCMEN1KMT2A
SCHEMBL8779760 0.77 ALDH1A1 (0.47) MEN1LMNAMAPTKMT2AALDH1A1
SCHEMBL8779758 0.77 ALDH1A1 (0.47) MEN1LMNAMAPTKMT2AALDH1A1
SCHEMBL8779675 0.72 MEN1 (0.57) MEN1LMNAPOLBMAPTKMT2A
SCHEMBL6848698 0.72 CYP2C9 (1.00) CYP2C9EEF2KSRCMEN1LMNA
SCHEMBL30682161 0.72 CYP2C9 (1.00) CYP2C9EEF2KSRCMEN1LMNA
SCHEMBL6851626 0.72 CYP2C9 (1.00) CYP2C9EEF2KSRCMEN1LMNA
SCHEMBL8779682 0.70 CYP1A2 (0.59) CYP2C9MEN1LMNAPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525197-B1 3-BENZYLIDENE-1-CARBAMOYL-2-PYRROLIDONE ANALOGS SHIONOGI & CO (JP) 1997-08-27 EP disclosed
US-5319100-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
US-5319099-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
EP-0525197-A1 3-BENZYLIDENE-1-CARBAMOYL-2-PYRROLIDONE ANALOG SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-02-03 EP disclosed