SCHEMBL8779758

SCHEMBL8779758

NC(=O)N1CC/C(=C/c2ccccc2)C1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
HTT P42858 1/20 0.47
CYP1A2 P05177 2/20 0.47
F3 P13726 1/20 0.45
ACHE P22303 1/20 0.42
MGAM O43451 3/20 0.42
GAA P10253 3/20 0.42
SI P14410 3/20 0.42
MGAM2 Q2M2H8 3/20 0.42
RCE1 Q9Y256 1/20 0.41
HDAC1 Q13547 4/20 0.40
MAPT P10636 3/20 0.40
RAB9A P51151 2/20 0.40
MEN1 O00255 1/20 0.40
MAPK1 P28482 1/20 0.40
MDM2 Q00987 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAOB P27338 2/20 0.40
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779760 1.00 ALDH1A1 (0.47) ALDH1A1HTTCYP1A2F3ACHE
SCHEMBL11332725 0.84 ALDH1A1 (0.47) ALDH1A1HTTCYP1A2F3ACHE
SCHEMBL11332739 0.84 ALDH1A1 (0.47) ALDH1A1HTTCYP1A2F3ACHE
SCHEMBL8779651 0.77 CYP2C9 (0.55) ALDH1A1HTTCYP1A2GAAMAPT
SCHEMBL8779657 0.77 CYP2C9 (0.55) ALDH1A1HTTCYP1A2GAAMAPT
SCHEMBL8779655 0.74 CYP1A2 (0.58) ALDH1A1CYP1A2GAAMEN1KMT2A
SCHEMBL8779659 0.74 CYP1A2 (0.58) ALDH1A1CYP1A2GAAMEN1KMT2A
SCHEMBL8779675 0.71 MEN1 (0.57) ALDH1A1HTTGAAMAPTRAB9A
SCHEMBL17161963 0.71 ACHE (0.68) ALDH1A1CYP1A2F3ACHEMGAM
SCHEMBL11325310 0.71 AKR1C3 (0.51) ALDH1A1CYP1A2ACHEHDAC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525197-B1 3-BENZYLIDENE-1-CARBAMOYL-2-PYRROLIDONE ANALOGS SHIONOGI & CO (JP) 1997-08-27 EP disclosed
US-5319100-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
US-5319100-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
US-5319100-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
US-5319099-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
US-5319099-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
US-5319099-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
EP-0525197-A1 3-BENZYLIDENE-1-CARBAMOYL-2-PYRROLIDONE ANALOG SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-02-03 EP disclosed
EP-0525197-A1 3-BENZYLIDENE-1-CARBAMOYL-2-PYRROLIDONE ANALOG SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-02-03 EP disclosed
WO-1992012966-A1 3-BENZYLIDENE-1-CARBAMOYL-2-PYRROLIDONE ANALOG SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1992-08-06 WO disclosed