SCHEMBL8779874

SCHEMBL8779874

C=C1CCCN1C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ESR2 Q92731 1/20 0.39
CTSK P43235 1/20 0.39
NR1H2 P55055 1/20 0.38
HPGD P15428 1/20 0.37
MPO P05164 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
EPHX1 P07099 1/20 0.36
BRD4 O60885 1/20 0.35
MAPK1 P28482 1/20 0.35
KDM1A O60341 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
PREP P48147 1/20 0.34
UCHL1 P09936 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5278772 0.95 HPGD (0.40) USP2SMN1; SMN2ESR2CTSKNR1H2
SCHEMBL1849006 0.93 HPGD (0.42) USP2SMN1; SMN2ESR2CTSKNR1H2
SCHEMBL27851257 0.89 USP2 (0.42) USP2SMN1; SMN2ESR2CTSKNR1H2
SCHEMBL13617428 0.81 ESR2 (0.37) USP2SMN1; SMN2ESR2CTSKNR1H2
SCHEMBL15188491 0.80 CTSK (0.44) USP2SMN1; SMN2ESR2CTSKNR1H2
SCHEMBL1550544 0.80 USP2 (0.41) USP2SMN1; SMN2ESR2CTSKNR1H2
SCHEMBL205421 0.80 LMNA (0.48) USP2SMN1; SMN2ESR2CTSKNR1H2
SCHEMBL7495565 0.79 LMNA (0.47) USP2SMN1; SMN2ESR2CTSKNR1H2
SCHEMBL16025271 0.79 USP2 (0.40) USP2SMN1; SMN2ESR2CTSKNR1H2
SCHEMBL4621580 0.79 USP2 (0.40) USP2SMN1; SMN2ESR2CTSKNR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773953-A1 COMBINATORIAL LIBRARIES OF MOLECULES AND METHODS FOR PRODUCING SAME THE SCRIPPS INSTITUTE (US) 1997-05-21 EP claimed
WO-1996003424-A1 COMBINATORIAL LIBRARIES OF MOLECULES AND METHODS FOR PRODUCING SAME THE SCRIPPS RESEARCH INSTITUTE (US) 1996-02-08 WO claimed
US-9834549-B2 3,3-disubstituted-(8-aza-bicyclo[3.2.1]OCT-8-yl)-[5-(1H-pyrazol-4-yl)-thiophen-3-yl]-methanones as inhibitors of 11 (β)-HSD1 THE UNIVERSITY OF EDINBURGH (GB) 2017-12-05 US disclosed
EP-2300469-B1 FUSED NITROGEN CONTAINING HETEROCYCLES AND COMPOSITIONS THEREOF AS KINASE INHIBITORS NOVARTIS AG (CH) 2015-06-24 EP disclosed