SCHEMBL8779999

SCHEMBL8779999

CS(=O)(=O)c1ccc(-c2ccccc2O)cc1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.69
ALDH1A1 P00352 1/20 0.54
HPGD P15428 1/20 0.54
BCL2L1 Q07817 1/20 0.54
HSD17B10 Q99714 1/20 0.54
DRD1 P21728 1/20 0.53
PTGS1 P23219 1/20 0.53
ADAMTS4 O75173 1/20 0.52
ENPP2 Q13822 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20590369 0.85 DRD1 (0.55) PTGS2ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL27516551 0.82 CA12 (0.65) PTGS2ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL6053300 0.82 ALDH1A1 (0.56) PTGS2ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL5502727 0.82 PTGS2 (1.00) PTGS2PTGS1
Hydrogen Sulfide SCHEMBL27744400 0.80 PTGS2 (0.96) PTGS2PTGS1
SCHEMBL387063 0.79 ENPP2 (0.61) PTGS2ENPP2
SCHEMBL20590368 0.79 DRD1 (0.58) PTGS2ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL6732777 0.78 PTGS2 (0.78) PTGS2DRD1
SCHEMBL714236 0.78 ALDH1A1 (0.83) ALDH1A1HPGDBCL2L1HSD17B10
SCHEMBL29443997 0.78 ALDH1A1 (0.83) ALDH1A1HPGDBCL2L1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102639500-B Tricyclic compound, preparation method and pharmaceutical use thereof SHANGHAI HENGRUI PHARM CO LTD 2015-02-11 CN disclosed
CN-102639500-A Tricyclic compound, preparation method and pharmaceutical use thereof SHANGHAI HENGRUI PHARM CO LTD 2012-08-15 CN disclosed
EP-0783486-A1 NOVEL PROSTAGLANDIN SYNTHASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-07-16 EP disclosed
US-5593994-A ANTIINFLAMMATORY AGENTS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-01-14 US disclosed