SCHEMBL8780449

SCHEMBL8780449

CCCCC1N=NC(=O)c2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
ALDH1A1 P00352 2/20 0.35
CYP3A4 P08684 2/20 0.35
GRM2 Q14416 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
PTGS1 P23219 1/20 0.35
RAB9A P51151 1/20 0.35
NAPRT Q6XQN6 1/20 0.35
AKT1 P31749 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21533082 0.83 MEN1 (0.36) BCHEACHEALDH1A1LMNACYP1A2
SCHEMBL8559782 0.81 TDO2 (0.38) ALDH1A1CYP3A4LMNACYP1A2CYP2C9
SCHEMBL11416663 0.77 MEN1 (0.36) ALDH1A1MAPTHPGD
SCHEMBL11412655 0.76 METAP1 (0.40)
SCHEMBL4213119 0.74 MAOB (0.39) ALDH1A1MAPT
SCHEMBL463373 0.73 APEX1 (0.39) ALDH1A1CYP1A2MAPT
SCHEMBL6474398 0.71 CYP19A1 (0.44) CYP3A4LMNACYP1A2CYP2C9TP53
SCHEMBL11817385 0.71 BCHE (0.37) BCHEACHEALDH1A1CYP3A4GRM2
SCHEMBL11411069 0.71 POLB (0.40) ACHEALDH1A1
SCHEMBL9482199 0.70 PTPRC (0.35) ALDH1A1CYP1A2TP53RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498722-B1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1997-07-30 EP claimed
EP-0498722-B1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1997-07-30 EP disclosed