SCHEMBL8780462

SCHEMBL8780462

CCCCc1cnc2ccccc2c1Cc1ccc(C#N)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 2/20 0.41
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.39
SMO Q99835 1/20 0.38
PDE10A Q9Y233 1/20 0.38
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLC22A12 Q96S37 1/20 0.36
CYP2A6 P11509 1/20 0.36
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
CYP19A1 P11511 3/20 0.35
TLR7 Q9NYK1 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118013 0.80 AGTR1 (0.47) TLR8TSHRALDH1A1SMN1; SMN2KDM4E
SCHEMBL8780493 0.80 TLR8 (0.42) TLR8TSHRHSD17B10SMOALDH1A1
SCHEMBL18554028 0.77 TLR8 (0.38) TLR8ABCG2SMOSLC22A12CYP2A6
SCHEMBL8675220 0.75 KDM4E (0.44) TLR8TSHRHSD17B10PDE10AALDH1A1
SCHEMBL8504620 0.75 BRS3 (0.54)
SCHEMBL8780501 0.75 MEN1 (0.42) TLR8TSHRHSD17B10ABCG2ALDH1A1
SCHEMBL9723340 0.74 PTPN1 (0.41) PDE10A
SCHEMBL18270667 0.74 TLR7 (0.51) TLR8HSD17B10ALDH1A1SMN1; SMN2KDM4E
SCHEMBL8501923 0.73 AGTR1 (0.50)
SCHEMBL27668508 0.69 TLR7 (0.47) TLR8TSHRHSD17B10ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4338378-A None JP disclosed
EP-0498722-B1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1997-07-30 EP disclosed
US-5478938-A Antagonists for angiotensin II receptors; hypotensive, cardiotonic agents; cognitive activators ROUSSEL UCLAF (FR) 1995-12-26 US disclosed
US-5324839-A Hypotensive agents, gastrointestinal and urogenital disorders ROUSSEL-UCLAF (FR) 1994-06-28 US disclosed
JP-H04338378-A NOVEL NITROGENOUS BICYCLIC DERIVATIVE SUBSTITUTED WITH BENZYL GROUP, THEIR PRODUCTION, RESULTED NOVEL INTERMEDIATE, ITS USE AS DRUG AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME ROUSSEL UCLAF 1992-11-25 JP disclosed
EP-0498722-A1 Bicyclic nitrogen compounds, their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1992-08-12 EP disclosed