SCHEMBL9723340

SCHEMBL9723340

CCCCc1cnc2ccccc2c1Cc1ccc(-c2ccccc2CC(=O)O)cc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.41
AGTR1 P30556 2/20 0.41
AGTR2 P50052 2/20 0.41
DHODH Q02127 1/20 0.41
LTB4R2 Q9NPC1 1/20 0.40
BRS3 P32247 2/20 0.40
PDE10A Q9Y233 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8504620 0.87 BRS3 (0.54) AGTR1AGTR2DHODHBRS3
SCHEMBL8501923 0.82 AGTR1 (0.50) AGTR1AGTR2LTB4R2BRS3
SCHEMBL9118013 0.82 AGTR1 (0.47) AGTR1AGTR2DHODH
SCHEMBL8780462 0.74 TLR8 (0.41) PDE10A
SCHEMBL9759625 0.74 ALDH1A1 (0.62) LTB4R2
SCHEMBL8675220 0.74 KDM4E (0.44) PDE10A
SCHEMBL7835618 0.71 BRS3 (0.52) AGTR1AGTR2DHODHLTB4R2BRS3
SCHEMBL7835619 0.70 PDE4A (0.41) AGTR1AGTR2DHODHBRS3PDE10A
SCHEMBL9654571 0.69 AGTR1 (0.56) AGTR1AGTR2DHODHLTB4R2
SCHEMBL28408449 0.68 PTGS1 (0.66)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4346974-A None JP disclosed
JP-H04346974-A NOVEL NITROGENOUS BICYCLIC DERIVATIVES, THEIR PRODUCTION, RESULTED NOVEL INTERMEDIATES, THEIR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME ROUSSEL UCLAF 1992-12-02 JP disclosed