SCHEMBL8780741

SCHEMBL8780741

Cc1noc(C)c1-c1nc(COc2ccc3cccc(N4CCN(C)CC4)c3c2)no1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.71
KCNH2 Q12809 1/20 0.71
HTR1A P08908 11/20 0.56
HTR1D P28221 10/20 0.56
HTR1B P28222 10/20 0.56
OPRL1 P41146 1/20 0.41
CYP1A2 P05177 4/20 0.40
ALDH1A1 P00352 4/20 0.40
USP2 O75604 1/20 0.40
TSHR P16473 3/20 0.40
LMNA P02545 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
MAPK1 P28482 2/20 0.40
CYP2D6 P10635 1/20 0.40
MTNR1B P49286 1/20 0.39
BRD4 O60885 1/20 0.39
CYP3A4 P08684 1/20 0.39
HIF1A Q16665 1/20 0.39
DRD2 P14416 1/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1387548 0.98 SLC6A9 (0.69) SLC6A9KCNH2HTR1AHTR1DHTR1B
SCHEMBL1387524 0.85 SLC6A9 (0.84) SLC6A9KCNH2HTR1AHTR1DHTR1B
SCHEMBL1387568 0.85 SLC6A9 (0.51) SLC6A9KCNH2HTR1AHTR1DHTR1B
Hydrochloric Acid SCHEMBL7813268 0.84 SLC6A9 (0.82) SLC6A9KCNH2HTR1AHTR1DHTR1B
SCHEMBL8185864 0.83 SLC6A9 (0.83) SLC6A9KCNH2HTR1AHTR1DHTR1B
SCHEMBL7813346 0.82 SLC6A9 (0.76) SLC6A9KCNH2HTR1AHTR1DHTR1B
Hydrochloric Acid SCHEMBL7810671 0.82 SLC6A9 (0.82) SLC6A9KCNH2HTR1AHTR1DHTR1B
SCHEMBL7803817 0.81 SLC6A9 (0.70) SLC6A9KCNH2HTR1AHTR1DHTR1B
Hydrochloric Acid SCHEMBL7813281 0.81 SLC6A9 (0.96) SLC6A9KCNH2HTR1AHTR1DHTR1B
Hydrochloric Acid SCHEMBL1387634 0.81 SLC6A9 (0.74) SLC6A9KCNH2HTR1AHTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795328-A1 Use of naphthalene derivatives in treating lung carcinoma PFIZER INC. (US) 1997-09-17 EP claimed
EP-0795328-A1 Use of naphthalene derivatives in treating lung carcinoma PFIZER INC. (US) 1997-09-17 EP disclosed