SCHEMBL8780938

SCHEMBL8780938

CCN(CCOc1ccc(-n2ccnc2)cc1)CCc1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 10/20 0.55
CYP2C9 P11712 10/20 0.55
CYP1A2 P05177 7/20 0.55
CYP2C19 P33261 6/20 0.55
CYP3A4 P08684 8/20 0.52
CYP19A1 P11511 1/20 0.52
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
KCNH2 Q12809 1/20 0.44
MCHR1 Q99705 1/20 0.44
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
GPR119 Q8TDV5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780823 0.94 CYP2D6 (0.53) CYP2D6CYP2C9CYP1A2CYP2C19CYP3A4
SCHEMBL8780782 0.89 CYP2D6 (0.54) CYP2D6CYP2C9CYP1A2CYP2C19CYP3A4
SCHEMBL8780902 0.85 CYP2D6 (0.56) CYP2D6CYP2C9CYP1A2CYP2C19CYP3A4
SCHEMBL8780791 0.83 CYP2D6 (0.51) CYP2D6CYP2C9CYP1A2CYP2C19CYP3A4
SCHEMBL8780940 0.81 ADORA2A (0.43) CYP2D6CYP2C9CYP1A2CYP2C19KCNH2
SCHEMBL7068561 0.81 CYP2D6 (0.77) CYP2D6CYP2C9CYP1A2CYP2C19CYP3A4
SCHEMBL10508102 0.79 CYP2D6 (0.70) CYP2D6CYP2C9CYP1A2CYP2C19CYP3A4
SCHEMBL8780777 0.78 KCNH2 (0.48) KCNH2MCHR1ADORA3ADORA2AADORA2B
SCHEMBL8780805 0.78 KCNH2 (0.65) KCNH2MCHR1ADORA3ADORA2AADORA2B
Hydrochloric Acid SCHEMBL10510793 0.78 CYP2D6 (0.68) CYP2D6CYP2C9CYP1A2CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed