SCHEMBL8780940

SCHEMBL8780940

CCN(CCOc1ccc(N)cc1)CCc1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.43
KCNH2 Q12809 2/20 0.43
ADORA1 P30542 2/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADORA2B P29275 1/20 0.43
MCHR1 Q99705 1/20 0.43
MAPT P10636 1/20 0.42
CHRNA7 P36544 1/20 0.42
KMT2A Q03164 1/20 0.42
SIGMAR1 Q99720 2/20 0.40
PKM P14618 1/20 0.39
EBP Q15125 1/20 0.39
TCF4 P15884 1/20 0.38
CTNNB1 P35222 1/20 0.38
CYP1A2 P05177 1/20 0.38
LTA4H P09960 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780789 0.93 ADORA2A (0.41) ADORA2AKCNH2ADORA1ADORA3ADORA2B
SCHEMBL8780815 0.92 ADORA2A (0.38) ADORA2AKCNH2ADORA1ADORA3ADORA2B
SCHEMBL8780919 0.90 HRH3 (0.41) ADORA2AKCNH2ADORA1ADORA3ADORA2B
SCHEMBL8780867 0.86 KCNH2 (0.43) ADORA2AKCNH2ADORA1ADORA3ADORA2B
SCHEMBL8780967 0.85 ADORA1 (0.39) KCNH2ADORA1MAPTKMT2ASIGMAR1
SCHEMBL8780776 0.85 MAOA (0.37) ADORA2AKCNH2ADORA1ADORA3ADORA2B
SCHEMBL8780805 0.84 KCNH2 (0.65) ADORA2AKCNH2ADORA1ADORA3ADORA2B
SCHEMBL8780777 0.83 KCNH2 (0.48) ADORA2AKCNH2ADORA1ADORA3ADORA2B
SCHEMBL8780824 0.83 TDP1 (0.39) ADORA2AKCNH2ADORA1ADORA3ADORA2B
SCHEMBL8780988 0.82 KCNH2 (0.41) KCNH2ADORA1MAPTKMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697407-B1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS (JP) 1997-06-25 EP disclosed
EP-0697407-A1 Pyrimidinedione derivatives and antiarrhythmic compositions containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-02-21 EP disclosed