SCHEMBL8780987

SCHEMBL8780987

CCCCCCCC(N)c1ccccc1OCc1ccccn1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
PPARG P37231 2/20 0.45
SYK P43405 8/20 0.43
TLR8 Q9NR97 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
AURKB Q96GD4 3/20 0.42
INCENP Q9NQS7 3/20 0.42
SLC1A5 Q15758 1/20 0.42
ABCB1 P08183 1/20 0.41
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
SLC2A1 P11166 1/20 0.39
GCK P35557 1/20 0.39
LPAR3 Q9UBY5 1/20 0.39
CYSLTR2 Q9NS75 1/20 0.38
CYSLTR1 Q9Y271 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8781026 0.99 CYP1A2 (0.47) CYP1A2PPARGSYKTLR8TLR7
SCHEMBL8781006 0.90 SYK (0.47) CYP1A2SYKTLR8TLR7AURKB
SCHEMBL8781190 0.86 CYP1A2 (0.44) CYP1A2PPARGSYKTLR8TLR7
SCHEMBL8780979 0.84 SYK (0.54) CYP1A2SYKTLR8TLR7AURKB
SCHEMBL8781114 0.79 SMO (0.43) CYP1A2SYKTLR8TLR7AURKB
SCHEMBL8781013 0.79 PDE4D (0.45) CYP1A2SYKAURKBINCENPSLC2A1
SCHEMBL8781040 0.79 SYK (0.45) SYKAURKBINCENPSLC2A1
SCHEMBL8780866 0.79 SLC2A1 (0.59) CYP1A2SYKTLR8TLR7AURKB
SCHEMBL462017 0.76 SIGMAR1 (0.50) PPARGSLC2A1CYSLTR2CYSLTR1
Hydrochloric Acid SCHEMBL10855754 0.76 SYK (0.41) CYP1A2PPARGSYKTLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773218-A1 N-(Piperazinylalkoxyphenyl)-N'phenylalkylurea derivatives as ACAT inhibitors for the treatment of atheroschlerosis MITSUBISHI CHEMICAL CORPORATION (JP) 1997-05-14 EP disclosed